A facile synthesis of optically pure amines by reduction of N-acyl-.ALPHA.-methoxyalkylamines derived from .ALPHA.-amino acids using triethylsilane.
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چکیده
منابع مشابه
One Pot Synthesis of Alpha-Aminonitrile and Alpha-Amino Acid From Schiff Bases
Addition of Potassium cyanide to a mixture of Schiff base and lithium perchlorate afforded a-aminonitriles in high yields. Addition of potassium cyanide to a methanolic solution of Schiff base and phosphoric acid afforded a-aminonitriles. When the reaction mixture was refluxed it gave a-amino acids in high yields.
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ژورنال
عنوان ژورنال: Chemical and Pharmaceutical Bulletin
سال: 1990
ISSN: 0009-2363,1347-5223
DOI: 10.1248/cpb.38.2024